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Structure-function of the G protein-coupled receptor superfamily

author

Vsevolod Katritch

2000 -

Raymond C Stevens

Vadim Cherezov

published in: Annual Review of Pharmacology and Toxicology

date of publication: 2012-11-08

main subject: G protein-coupled receptor

Cites articles 117

Date

Title

Authors

2012-07-13

Structural Basis for Allosteric Regulation of GPCRs by Sodium Ions

Vsevolod Katritch, Vadim Cherezov, Laura H Heitman, Adriaan P IJzerman, Raymond C Stevens, Gye Won Han, Pavel Chubukov
2012-05-16

Structure of the δ-opioid receptor bound to naltrindole

William I Weis, Brian Kobilka, Aashish Manglik, Tong Sun Kobilka
2012-05-16

Structure of the nociceptin/orphanin FQ receptor in complex with a peptide mimetic

Vsevolod Katritch, Vadim Cherezov, Huixian Wu, Xi-Ping Huang, Claudio Trapella, Remo Guerrini, Bryan L. Roth, Raymond C Stevens, Eyal Vardy, Girolamo Calò
2012-05-09

Crystal Structures of a Stabilized β1-Adrenoceptor Bound to the Biased Agonists Bucindolol and Carvedilol

Tony Warne, Christopher G. Tate
2012-04-09

Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy
2012-04-30

Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening

Vsevolod Katritch, Ruben Abagyan, Kenneth A. Jacobson, Zhan-Guo Gao, Dilip K Tosh, Raymond C Stevens, Francesca Deflorian
2012-05-17

Structure of the human κ-opioid receptor in complex with JDTic

Vsevolod Katritch, Vadim Cherezov, Daniel Wacker, Huixian Wu, Xi-Ping Huang, Bryan L. Roth, Raymond C Stevens, Gye Won Han, Eyal Vardy, F. Ivy Carroll, Richard B Westkaemper, Philip D Mosier
2012-03-21

Crystal structure of the µ-opioid receptor bound to a morphinan antagonist

Jesper M Mathiesen, Leonardo Pardo, William I Weis, Brian Kobilka, Aashish Manglik, Tong Sun Kobilka
2012-03-19

Structure-based ligand discovery for the protein-protein interface of chemokine receptor CXCR4

Dahlia R Weiss, Nikolaus Heveker
2012-02-22

Structure and dynamics of the M3 muscarinic acetylcholine receptor

Erica Rosemond, Albert C Pan, William I Weis, Brian Kobilka, Pil Seok Chae, Ron Ofer Dror
2012-02-17

Crystal structure of a lipid G protein-coupled receptor

Raymond C Stevens
2012-01-29

G-protein-coupled receptor inactivation by an allosteric inverse-agonist antibody

Takatoshi Arakawa, Alexander Cameron, Takeshi Murata
2012-02-23

Structure of the human M2 muscarinic acetylcholine receptor bound to an antagonist

Cheng Zhang, William I Weis, Brian Kobilka, Hidetsugu Asada
2012-01-19

Biased signaling pathways in β2-adrenergic receptor characterized by 19F-NMR.

Vsevolod Katritch, Raymond C Stevens, Reto Horst, Kurt Wüthrich
2012-03-08

Discovery of 1,2,4-Triazine Derivatives as Adenosine A 2A Antagonists using Structure Based Drug Design

Christopher J Langmead
2012-01-03

Stabilized G protein binding site in the structure of constitutively active metarhodopsin-II

Jörg Standfuss, Xavier Deupí, Gebhard Schertler
2012-01

Diversity and modularity of G protein-coupled receptor structures

Vsevolod Katritch, Vadim Cherezov, Raymond C Stevens
2012-03-01

Lifting the lid on GPCRs: the role of extracellular loops

David R Poyner, Denise Wootten, Mark Wheatley, John Simms
2011-12-08

Crystal structure-based virtual screening for fragment-like ligands of the human histamine H(1) receptor

Vsevolod Katritch, Albert Kooistra, Chris de Graaf
2011-09-28

Conformational changes in the G protein Gs induced by the β2 adrenergic receptor

Ka Young Chung, Søren G. F. Rasmussen, Brian T Devree, Brian Kobilka
2011-09-19

Molecular mechanism of β-arrestin-biased agonism at seven-transmembrane receptors

Arun K Shukla, Robert Lefkowitz
2011-10-21

Conformational dynamics of single G protein-coupled receptors in solution

Brian Kobilka, Alexandre Fürstenberg, William E. Moerner
2011-09-18

Ligand discovery from a dopamine D3 receptor homology model and crystal structure

John J Irwin, Brian K. Shoichet, Avner Schlessinger, Andrej Šali, Ryan G Coleman, Jens Carlsson, Bryan L. Roth, Avner Schlessinger
2011-09-09

The best of both worlds? Bitopic orthosteric/allosteric ligands of g protein-coupled receptors
2011-09-01

Ligand-dependent perturbation of the conformational ensemble for the GPCR β2 adrenergic receptor revealed by HDX.

Vsevolod Katritch
2011-09-07

Structure of the Adenosine A2A Receptor in Complex with ZM241385 and the Xanthines XAC and Caffeine

Nathan Robertson, Francesca Magnani, Fiona H. Marshall, Christopher G. Tate
2011-01-01

Oligomerization of G protein-coupled receptors: computational methods
2011-01-01

Oligomerization of G protein-coupled receptors: biochemical and biophysical methods

Agnieszka Kaczor
2011-08-01

Status of GPCR modeling and docking as reflected by community-wide GPCR Dock 2010 assessment

Irina Kufareva, Vsevolod Katritch, Ruben Abagyan
2011-07-21

Pathway and mechanism of drug binding to G-protein-coupled receptors

David W. Borhani, Huafeng Xu, Ron Ofer Dror
2011-09-29

Crystal structure of the β2 adrenergic receptor-Gs protein complex

Jan Steyaert, Els Pardon, Joseph A Lyons, Martin Caffrey, William I Weis, Jesper M Mathiesen, Georgios Skiniotis, Brian Kobilka, Tong Sun Kobilka, Pil Seok Chae, Søren G. F. Rasmussen, Roger K Sunahara, Foon Sun Thian, Samuel H. Gellman, Yaozhong Zou
2011-06-29

Structural insights into RAMP modification of secretin family G protein-coupled receptors: implications for drug development

Debbie Hay, Joseph Gingell, Julia K Archbold

Article - wd:Q30576993

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