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Discovery of Nonstandard Macrocyclic Peptides as Noncompetitive Inhibitors of the Zika Virus NS2B-NS3 Protease

author

Toby Passioura

Christian Klein

2000 -

Hiroaki Suga

1963 -

Gottfried Otting

published in: ACS Medicinal Chemistry Letters

date of publication: 2019-01-04

language: English

main subject: Zika virus

Cites articles 29

Date

Title

Authors

2018-01-25

Development of vaccines against Zika virus.

Gregory A. Poland, Inna G Ovsyannikova, Jorge Elias Kalil Filho
2018-04-30

Cyclization of peptides with two chemical bridges affords large scaffold diversities

Xu-Dong Kong, Christian Heinis
2018-05-17

De Novo Macrocyclic Peptide Inhibitors of Hepatitis B Virus Cellular Entry

Toby Passioura, Masashi Mizokami, Yasuhito Tanaka, Takaji Wakita, Koichi Watashi
2018-10-10

Structures of Zika virus NS2B-NS3 protease in complex with peptidomimetic inhibitors

Dahai Luo, Zhenzhen Zhang
2017-02-01

Highly Constrained Bicyclic Scaffolds for the Discovery of Protease-Stable Peptides via mRNA Display

Teresa M. Przytycka, Emil S Iqbal, Matthew C T Hartman
2017-02-16

Rapid Discovery of Potent and Selective Glycosidase-Inhibiting De Novo Peptides
2017-04-29

Characterization of the Zika virus two-component NS2B-NS3 protease and structure-assisted identification of allosteric small-molecule antagonists

Sujan Shresta, Annie Elong Ngono, Alexey V Terskikh
2017-05-25

A conformational switch high-throughput screening assay and allosteric inhibition of the flavivirus NS2B-NS3 protease

Matthew Brecher, Adham Alifarag, Laura D Kramer, Hongmin Li
2017-06-02

Macrocyclic peptide inhibitors for the protein-protein interaction of Zaire Ebola virus protein 24 and karyopherin alpha 5.

Toby Passioura, Hiroaki Suga
2017-06-21

An update on Zika virus infection

Didier Musso, Duane J. Gubler, David Baud, Marion C. Lanteri, Bruno Schaub
2017-06-23

Structural Dynamics of Zika Virus NS2B-NS3 Protease Binding to Dipeptide Inhibitors

Yan Li, Shuang Liu, CongBao Kang, Dahai Luo, Zhenzhen Zhang
2017-07-10

Solution conformations of Zika NS2B-NS3pro and its inhibition by natural products from edible plants

Jianxing Song
2016-04-14

Development of Potent and Selective S. aureus Sortase A Inhibitors Based on Peptide Macrocycles

Shawna McCallin
2016-07-07

Crystal structure of Zika virus NS2B-NS3 protease in complex with a boronate inhibitor

Rolf Hilgenfeld, Christian Klein
2016-11-15

Structure of the NS2B-NS3 protease from Zika virus after self-cleavage

Julien Lescar, Dahai Luo, Yan Li, CongBao Kang, Zhenzhen Zhang
2016-12-08

Crystal structure of unlinked NS2B-NS3 protease from Zika virus

Yan Li, CongBao Kang, Dahai Luo
2016-12-14

Peptide-Boronic Acid Inhibitors of Flaviviral Proteases: Medicinal Chemistry and Structural Biology

Christian Klein, Ralf Bartenschlager, Rolf Hilgenfeld
2016-10-27

Allosteric Inhibition of a Semaphorin 4D Receptor Plexin B1 by a High-Affinity Macrocyclic Peptide.

Yu Kitago
2015-09-14

Phenylalanine and Phenylglycine Analogues as Arginine Mimetics in Dengue Protease Inhibitors

Christian Klein, Ralf Bartenschlager
2014-02-21

Selection-based discovery of druglike macrocyclic peptides

Toby Passioura, Takayuki Katoh
2014-09-30

Biochemistry and medicinal chemistry of the dengue virus protease

Christian Klein, Tanja Schirmeister
2014-12-08

Novel dengue virus NS2B/NS3 protease inhibitors

Jochen Bodem, Tanja Schirmeister, Ralf Bartenschlager
2013-10-22

Thiazolidinone-peptide hybrids as dengue virus protease inhibitors with antiviral activity in cell culture

Christian Klein, Mira A M Behnam, Anil Kumar, Ralf Bartenschlager
2013-12-20

Allosteric Inhibition of the NS2B-NS3 Protease from Dengue Virus
2012-02-26

Retro peptide-hybrids as selective inhibitors of the Dengue virus NS2B-NS3 protease

Christian Steuer, Christian Klein, Mira A M Behnam
2011-12-01

Natural product-like macrocyclic N-methyl-peptide inhibitors against a ubiquitin ligase uncovered from a ribosome-expressed de novo library

Takayuki Katoh
2008-01-24

Reprogramming the translation initiation for the synthesis of physiologically stable cyclic peptides
2007-12

The design of drugs for HIV and HCV

Erik De Clercq
1974-01

A simple graphical method for determining the inhibition constants of mixed, uncompetitive and non-competitive inhibitors

Article - wd:Q61795450

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